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University of Groningen Carbon-carbon bond formations using organolithium reagents Heijnen, Dorus

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University of Groningen

Carbon-carbon bond formations using organolithium reagents

Heijnen, Dorus

IMPORTANT NOTE: You are advised to consult the publisher's version (publisher's PDF) if you wish to cite from it. Please check the document version below.

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Publication date: 2018

Link to publication in University of Groningen/UMCG research database

Citation for published version (APA):

Heijnen, D. (2018). Carbon-carbon bond formations using organolithium reagents. University of Groningen.

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List of publications

1) Gottumukkala, A. L.; Teichert, J.F.; Ferrer, C.; Eisink, N.; Heijnen, D.; van Dijk, S.; van

den Hoogenband, A.; Minnaard, A. J.

Pd-Diimine: A Highly Selective Catalyst System for the

Base-Free Oxidative Heck Reaction

J. Org. Chem. 2011,76, 3498.

2) Martín Fañanás-Mastral, Johannes F. Teichert, José Fernández, Dorus Heijnen, Ben L. Feringa.

Enantioselective synthesis of almorexant via iridium-catalysed intramolecular allylic

amidation Org. Biomol. Chem.

, 2013,

11

, 4521-4525

3) Alexander J. Cresswell , Stephen G. Davies, Aude L. A. Figuccia, Ai M. Fletcher, Dorus Heijnen, James A. Lee, Melloney J. Morris, Alice M. R. Kennett, Paul M. Roberts, James E. Thomson.

Pinacolatoboron fluoride (pinBF) is an efficient fluoride transfer agent for

diastereoselective synthesis of benzylic fluorides

Tetrahedron Letters. 2015, 56, 3373–3377 4) Dorus Heijnen, Valentín Hornillos, Brian P. Corbet, Massimo Giannerini, Ben L. Feringa.

Palladium-Catalyzed C(sp

3

)–C(sp

2

) Cross-Coupling of (Trimethylsilyl)methyllithium with

(Hetero)Aryl Halides

Org. Lett., 2015, 17 (9), 2262–2265

5) Jeffrey Buter, Dorus Heijnen, Carlos Vila,Valentin Hornillos,Edwin Otten, Massimo Giannerini, Adriaan J. Minnaard, Ben L. Feringa. Palladium-Catalyzed,

tert-

Butyllithium-Mediated

Dimerization of Aryl Halides and Its Application in the Atropselective Total Synthesis of Mastigophorene A

Angew.Chem .Int. Ed. 2016, 55,3620 –3624

6)

Dorus Heijnen, Jean-Baptiste Gualtierotti, Valentin Hornillos, Ben L. Feringa.

Nickel-Catalyzed Cross-Coupling of Organolithium Reagents with (Hetero)Aryl Electrophiles Chem. Eur. J. 2016, 22, 3991–3995

7) Wolters, Alexander T.; Hornillos, Valentin; Heijnen, Dorus; Giannerini, Massimo; Feringa, Ben L.

One-Pot, Modular Approach to Functionalized Ketones via Nucleophilic Addition of

Alkyllithium Reagents to Benzamides and Pd-Catalyzed α-Arylation.

ACS Catal., 2016, 6, 2622-2625

8)

Jeffrey Buter, Dorus Heijnen, Ieng Chim Wan, F. Matthias Bickelhaupt, David C. Young, Edwin Otten, D. Branch Moody, Adriaan J. Minnaard.

Stereoselective Synthesis of 1-Tuberculosinyl

Adenosine; a Virulence Factor of Mycobacterium tuberculosis

J. Org. Chem. 2016, 81, 6686−6696

9) Dorus Heijnen,Filippo Tosi,Carlos Vila, Marc C. A. Stuart, Philip H. Elsinga,Wiktor Szymanski, and Ben L. Feringa Oxygen Activated, Palladium Nanoparticle Catalyzed, Ultrafast Cross-Coupling of Organolithium Reagents

Angew.Chem. Int. Ed. 2017, 56,3354 –3359

10) Narayan Sinha, Dorus Heijnen,Ben L. Feringa, Micheal G. Organ. The cross-coupling of organolithium reagents at cryogenic temperatures; a one-pot procedure for the sequential coupling of C-, S-, and N-nucleophiles -submitted-

11) Dorus Heijnen, Milan van Zuylen, Filippo Tosi, Ben L Feringa, The cross coupling of carbolithiated acetylenes, and the synthesis of Z-Tamoxifen -Manuscript in preparation-

12) Dorus Heijnen, Hugo Helbert, Ben L. Feringa, The synthesis of substituted benzaldehydes via a one pot reduction/cross coupling procedure -Manuscript in preparation-

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13) Hugo Helbert, Jorn, Dorus Heijnen, Ben L. Feringa. One pot strategies for the synthesis of substituted keto-anilines -Manuscript in preparation-

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